| 1 |
Renin inhibitors: A paradigm for the design of orally active peptide-based therapeutic agents
Pages 1 -
13
Saul H. Rosenberg
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| 2 |
Analgesic effects of synthetic TRP (NPS) - containing dipeptides and analogues
Pages 15 -
32
M. T. García-López, R. Herranz, R. González-Muñiz, J. Del Río
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| 3 |
Design of RNA interactive anti-HIV-1 agents
Pages 33 -
41
Lucjan Strekowski, W. David Wilson, David W. Boykin, Raymond F. Schinazi, Jerzy L. Mokrosz
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| 4 |
Polyamines: A case of multiple yet specific receptor recognition
Pages 43 -
65
Carlo Melchiorre, Maurizio Recanatini, Maria L. Bolognesi, Paola Filippi, Anna Minarini
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| 5 |
Structure-activity relationships of acetylcholinesterase inhibitor: 1-benzyl-4-[(5, 6-dimethoxy-1-indanon-2-yl) methyl] piperidine hydrochloride (E2020) and related compounds
Pages 67 -
81
Hachiro Sugimoto
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| 6 |
A new generation of 1, 4-dihydropyridines showing novel pharmacological properties
Pages 83 -
91
M. P. Ortega, C. E. Sunkel, M. M. Gómez, L. Santons, M. Fau de Casa-Juana, J. G. Priego
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| 7 |
Aspects of antibody directed enzyme prodrug therapy (ADEPT)
Pages 93 -
100
C. J. Springer
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| 8 |
The structure-activity relationships of dibenz (c,e) azocines and 4-phenyl - 1,2,3,4-tetrahydroisoquinolin-4-ols as α-adrenergic blocking agents and noradrenaline potentiators
Pages 101 -
113
Masaru Kihara
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| 9 |
Studies on the α-adrenergic receptor: Structure-activity relationships
Pages 115 -
127
Gloria Resell, Mercedes Alvarez
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| 10 |
Novel 4-regiomodified anilidopiperidines. New analgesics with diverse profiles: Their development and therapeutic potential
Pages 129 -
143
Jerome R. Bagley, Linas V. Kudzma
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| 11 |
Some aspects of the structure-activity relationships in oxytocin and vasopressin
Pages 145 -
154
M. Tarnowska, A. Liwo, F. Kasprzykowski, L. Lankiewicz, Z. Grzonka, J. Ciarkowski
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| 12 |
NMR spectroscopy and drug metabolism: Studies of cyclophosphamide metabolites
Pages 155 -
171
Susan M. Ludeman, Gerald Zon, O. Michael Colvin, Michael P. Gamcsik, Ellen M. Shulman - Roskes
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| 13 |
A novel approach to the development of safer anti-inflammatory steroids: Antedrug
Pages 173 -
202
Mounir A. Khalil, Taesoo Kwon, Henry J. Lee
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| 14 |
Development of boron containing pyrimidine and nucleoside analogues for neutron capture therapy
Pages 203 -
221
Naganna M. Goudgaon, Raymond F. Schinazi
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| 15 |
A decade of 7-oxabicycloheptanes
Pages 223 -
241
Steven E. Hall
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| 16 |
Development of high-affinity ligands for serotonin receptor subtypes
Pages 243 -
260
I. van Wijngaarden, M. Th. M. Tulp, W. Soudijn
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| 17 |
14-Alkoxymorphinans-a series of highly potent opioid agonists, antagonists, and partial agonists
Pages 261 -
276
Helmut Schmidhammer
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| 18 |
A working hypothesis to explain the mechanism of action of gastrin
Pages 277 -
289
Jean Martinez, Jean-Claude Galleyrand, Jean Christophe Lallement, Muriel Amblard
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| 19 |
Potassium channel activators and airway function
Pages 291 -
311
D. R. Buckle, D. G. Smith
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| 20 |
The carbonic anhydrases: Are these enzymes still a good deal for a pharmacologist?
Pages 313 -
347
Francesco Botrè, Claudio Botrè
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| 21 |
Potential targets of anti-HIV drugs
Pages 349 -
357
Mohamed Nasr, Steven R. Turk
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| 22 |
Semisynthetic dalbaheptides: Chemistry and biological activity
Pages 359 -
376
Adriano Malabarba, Romeo Ciabatti, Bruno Cavalleri
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| 23 |
Stereoselectivity of excitatory amino acid receptors: Enzymatic resolution of AMPA receptor agonists
Pages 377 -
385
Jan J. Hansen
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| 24 |
Kadsurenone and 2,5-diaryl tetrahydrofurans PAF-receptor antagonists
Pages 387 -
425
Mitree M. Ponpipom
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| 25 |
Inhibition of calcification of costal cartilage by α-amino acids, simple peptides, and sulfur - containing compounds
Pages 427 -
437
William O. Foye, Anna W. Tai, Hwi Shin Chun
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| 26 |
Discovery of a potent, selective and orally active series of peptide leukotriene antagonists: Evolution of ICI 204.219
Pages 439 -
451
Ying Kwong Yee
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| 27 |
Separation of electronic, hydrophobic, and steric effects in 3D-quantitative structure-activity relationships with descriptors directly from 3D structures using a comparative molecular field analysis (CoMFA) approach
Pages 453 -
467
Ki Hwan Kim
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